Transition-metal-free cross-coupling of thioethers with aryl(cyano)iodonium triflates: a facile and efficient method for the one-pot synthesis of thiocyanates.

نویسندگان

  • Dan Zhu
  • Denghu Chang
  • Lei Shi
چکیده

A novel transition-metal-free cross-coupling method for the one-step synthesis of thiocyanates via the C-S bond cleavage of readily available thioethers with aryl(cyano)-iodonium triflates as the cyanating agent is developed. This process features relatively broad substrate scopes, less-toxic hypervalent iodine reagents, mild operating conditions, excellent functional group compatibilities, and affords various thiocyanates in moderate to good yields.

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عنوان ژورنال:
  • Chemical communications

دوره 51 33  شماره 

صفحات  -

تاریخ انتشار 2015